Estrano[17,16-e]pyrimidine-peptide conjugates

Tomohiro Matsumoto, Masataka Watanabe, Shuntaro Mataka, Thies Thiemann

Research output: Contribution to journalArticlepeer-review

18 Citations (Scopus)


The preparation of a steroidal heterocycle linked to the tripeptide Cys-Gly-Cys is described. Initially, an estrane-derived steroidal heterocycle containing an aminopyrimidine ring fused to the 16,17-position of the steroidal nucleus was synthesized. Thereafter, protected amino acids were coupled iteratively by the DCC method, commencing at the amino group of the aminopyrimidine unit.

Original languageEnglish
Pages (from-to)751-757
Number of pages7
Issue number9
Publication statusPublished - Oct 2003
Externally publishedYes


  • Estranes
  • Fused steroids
  • Peptides
  • Pyrimidines
  • Synthesis

ASJC Scopus subject areas

  • Biochemistry
  • Molecular Biology
  • Endocrinology
  • Pharmacology
  • Clinical Biochemistry
  • Organic Chemistry


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